Publications

  • Journal Papers

77. Wei-Yi Ding, Peiyuan Yu, Qian-Jin An, Katherine L. Bay, Shao-Hua Xiang, Shaoyu Li, Ying Chen, K.N. Houk*, Bin Tan*. DFT-guided phosphoric-acid-catalyzed atroposelective arene functionalization of nitrosonaphthalene. Chem. 2020, doi.org/10.1016/j.chempr.2020.06.001

76. Ye-Hui Chen#, Heng-Hui Li#, Xiao Zhang, Shao-Hua Xiang,* Shaoyu Li, Bin Tan*. Organocatalytic enantioselective synthesis of atropisomeric aryl-p-quinones: Platform molecules for diversity-oriented synthesis of biaryldiols. Angew. Chem. Int. Ed. 2020, doi.org/10.1002/anie.202004671

75. Shengyi Yan, Wang Xia, Shaoyu Li, Qiuling Song*, Shao-Hua Xiang, Bin Tan*. Michael reaction inspired atroposelective construction of axially chiral biaryls. J. Am. Chem. Soc. 2020142, 7322.

74. Wang Xia, Qian-Jin An, Shao-Hua Xiang, Shaoyu Li, Yong-Bin Wang, Bin Tan*. Chiral phosphoric acid catalyzed atroposelective C-H amination of arenes. Angew. Chem. Int. Ed. 202059, 6775.

73. Jian Zhang, Yi-Yan Wang, He Sun, Shao-Yu Li, Shao-Hua Xiang, Bin Tan*. Enantioselective three-component Ugi reaction catalyzed by chiral phosphoric acid. Sci.China Chem. 202063, 47.

72. Yong-Bin Wang, Quan-Hao Wu,  Zhi-Peng Zhou, Shao-Hua Xiang,  Yuan Cui, Peiyuan Yu, Bin Tan*. Asymmetric construction of axially chiral 2-arylpyrroles by chirality transfer of atropisomeric alkenes. Angew. Chem. Int. Ed. 201958, 13443.

71. Shuai Zhu, Ye-Hui Chen, Yong-Bin Wang, Peiyuan Yu, Shao-Yu Li, Shao-Hua Xiang, Jun-Qi Wang, Jian Xiao, Bin Tan*. Organocatalytic atroposelective construction of axially chiral arylquinones. Nat. Commun. 201910, 4268.

70. Dong-Liang Lu, Ye-Hui Chen, Shao-Hua Xiang, Peiyuan Yu, Bin Tan, Shaoyu Li*. Atroposelective construction of arylindoles by chiral phosphoric acid-catalyzed cross-coupling of indoles and quinones. Org. Lett. 201921, 6000.

69. Yong-Bin Wang, Peiyuan Yu, Zhi-Peng Zhou, Jian Zhang, Jun (Joelle) Wang, Shi-Hui Luo, Qiang-Shuai Gu, K. N. Houk*, Bin Tan*. Rational design, enantioselective synthesis and catalytic applications of axially chiral EBINOLs. Nat. Catal. 20192, 504. 

68. Liang-Wen Qi, Shaoyu Li, Shao-Hua Xiang, Jun (Joelle) Wang*, Bin Tan*. Asymmetric construction of atropisomeric biaryls via a redox neutral cross-coupling strategy. Nat. Catal. 20192, 314. 

67. Lei Zhang, Shao-Hua Xiang, Jun (Joelle) Wang*, Jian Xiao, Jun-Qi Wang, Bin Tan*. Phosphoric acid-catalyzed atroposelective construction of axially chiral arylpyrroles. Nat. Commun. 201910, 566.

66. Lin-Lin Zhang, Bing-Chao Da, Shao-Hua Xiang*, Shuai Zhu, Zi-Yun Yuan, Zhen Guo*, Bin Tan*.  Organocatalytic double arylation of 3-isothiocyanato oxindoles: Stereocontrolled synthesis of complex spirooxindoles. Tetrahedron 201975, 1689.

65. Lin-Lin Zhang, Ji-Wei Zhang, Shao-Hua Xiang*, Zhen Guo*, Bin Tan*. Stereoselective construction of complex spirooxindoles via bisthiourea catalyzed three-component reactions. Chin. J. Chem. 201836, 1182.

64. Lin-Lin Zhang, Ji-Wei Zhang, Shao-Hua Xiang*, Zhen Guo*, Bin Tan*. Remote control of axial chirality: Synthesis of spirooxindole–urazoles via desymmetrization of ATAD. Org. Lett. 201820, 6022.

63. Jian Zhang, Peiyuan Yu, Shao-Yu Li, He Sun, Shao-Hua Xiang,Jun (Joelle) Wang, Kendall N. Houk*, Bin Tan*. Asymmetric phosphoric acid–catalyzed four-component Ugi reaction. Science 2018361, eaas8708.

62. Yong-Bin Wang, Bin Tan*. Construction of Axially Chiral Compounds via Asymmetric Organocatalysis. Acc. Chem. Res. 201851, 534.

61. Xiao Zhang, Ye-Hui Chen, Bin Tan*. Organocatalytic enantioselective transformations involving quinone derivatives as reaction partners. Tetrahedron Lett.201859, 473. 

60. Liang-Wen Qi, Jian-Hui Mao, Jian Zhang and Bin Tan*. Organocatalytic Asymmetric Arylation of Indoles Enabled by Azo Groups. Nat. Chem. 201810, 58. 

59. Ye-Hui Chen, Liang-Wen Qi, Fang Fang, and Bin Tan*. Organocatalytic Atroposelective Arylation of 2-Naphthylamines as a Practical Approach to Axially Chiral Biaryl Amino Alcohols. Angew. Chem. Int. Ed. 201756, 16308.  

58. Yong-Bin Wang, Sheng-Cai Zheng, Yu-Mei Hu and Bin Tan*. Brønsted Acid-Catalysed Enantio-selective Construction of Axially Chiral Arylquinazolinones. Nat. Commun. 20178, 15489.

57. Sheng-Cai Zheng, San Wu, Yun-Hao Zhang, Qinghai Zhou, Lung Wa Chung, Liu Ye and Bin Tan*. Organocatalytic Atroposelective Synthesis of Axially Chiral Styrenes. Nat. Commun. 20178, 15238.

56. Lei Zhang, Jian Zhang, Ji Ma, Dao-Juan Cheng and Bin Tan*. Highly Atroposelective Synthesis of Arylpyrroles by Catalytic Asymmetric Paal-Knorr Reaction. J. Am. Chem. Soc. 2017139, 1714.

55. Jin-Shun Lin, Xiao-Yang Dong, Tao-Tao Li, Na-Chuan Jiang, Bin Tan, and Xin-Yuan Liu*. A Dual-Catalytic Strategy To Direct Asymmetric Radical Aminotrifluoromethylation of Alkenes. J. Am. Chem. Soc. 2016138, 9357.

54. Jin-Hui Xu, Sheng-Cai Zheng, Ji-Wei Zhang, Xin-Yuan Liu, and Bin Tan*. Construction of Tropane Derivatives by Organocatalytic Asymmetric Dearomatization of Isoquinolines. Angew. Chem. Int. Ed. 201655, 11834–11839. 

53. Xiao-Long Yu, Liping Kuang, Su Chen, Xiao-Long Zhu, Zhong-Liang Li, Bin Tan, and Xin-Yuan Liu,* Counteranion-Controlled Unprecedented Diastereo- and Enantioselective Tandem Povarov Reaction for Construction of Bioactive Octahydro-dipyrroloquinolines. ACS Catal. 2016, 6, 6182.

52. Ji-Wei Zhang, Jin-Hui Xu, Dao-Juan Cheng, Chuan Shi, Xin-Yuan Liu* and Bin Tan*. Discovery and Enantiocontrol of Axially Chiral Urazoles via Organocatalytic Tyrosine Click Reaction. Nat. Commun. 20167, 10677.

51. Can-Liang Ma, Xiao-Hua Li, Xiao-Long Yu, Xiao-Long Zhu, Yong-Zhou Hu, Xiao-Wu Dong,* Bin Tan,* and Xin-Yuan Liu*. Gold-catalyzed tandem synthesis of bioactive spiro-dipyrroloquinolines and its application in the one-step synthesis of incargranine B aglycone and seneciobipyrrolidine (I). Org. Chem. Front. 2016,3, 324.

50. Ning-Yuan Yang, Zhong-Liang Li, Liu Ye, Bin Tan, and Xin-Yuan Liu*. Organic base-catalysed solvent-tuned chemoselective carbotrifluoromethylation and oxytrifluoromethylation of unactivated alkenes. Chem. Commun. 201652, 9052.

49. Shao-Yu Li, Ji-Wei Zhang, Xian-Lin Li, Dao-Juan Cheng,and Bin Tan*. Phosphoric Acid-Catalyzed Asymmetric Synthesis of SPINOL Derivatives. J. Am. Chem. Soc. 2016138, 16561.

48. Lei Li, Zhong-Liang Li, Fu-Li Wang, Zhen Guo, Yong-Feng Cheng, Na Wang, Chao Fang, Jingjiang Liu, Chunhui Hou, Bin Tan, and Xin-Yuan Liu*. Radical Aryl Migration Enables Diversity-Oriented Synthesis of Structurally Diverse Medium/Macro- or Bridged-Rings. Nat. Commun. 20167, 13852.

47. Lin Huang, Jin-Shun Lin, Bin Tan,* Xin-Yuan Liu*. Alkene Trifluoromethylation-Initiated Remote α-Azidation of Carbonyl Compounds toward Trifluoromethyl γ-Lactam and Spirobenzofuranone-lactam. ACS Catal. 20155, 2826.

46. Ming-Yue Wu, Wei-Wei He, Xin-Yuan Liu*, Bin Tan*. Asymmetric Construction of Spirooxindoles by Organocatalytic Multicomponent Reactions Using Diazooxindoles. Angew. Chem. Int. Ed. 201554, 9409.

45. Zhi-Jia Fang, Sheng-Cai Zheng, Zhen Guo, Jing-Yao Guo, Bin Tan,* and Xin-Yuan Liu*. Asymmetric Synthesis of Axially Chiral Isoquinolones: Nickel-Catalyzed Denitrogenative Transannulation. Angew. Chem. Int. Ed. 201554, 9528.

44. Ye-Hui Chen,Dao-Juan Cheng,Jian Zhang,Yong Wang,Xin-Yuan Liu*, and Bin Tan*.Atroposelective Synthesis of Axially Chiral Biaryldiols via Organocatalytic Arylation of 2‑Naphthols. J. Am. Chem. Soc. 2015137, 15062.

43. Jin-Shun Lin, Peng Yu, Lin Huang, Pan Zhang, Bin Tan,* and Xin-Yuan Liu*. Brønsted Acid-Catalyzed Asymmetric Hydroamination of Alkenes: Synthesis of Pyrrolidines Bearing a Tetrasubstituted Carbon Stereocenter. Angew. Chem. Int. Ed. 201554, 7847.

42. Lin Huang, Sheng-Cai Zheng, Bin Tan,* Xin-Yuan Liu.* Metal-Free Direct 1,6- and 1,2-Difunctionalization Triggered by Radical Trifluoromethylation of Alkenes. Org. Lett. 201517, 1589.

41. Peng Yu, Sheng-Cai Zheng, Ning-Yuan Yang, Bin Tan,* and Xin-Yuan Liu.* Phosphine-Catalyzed Remote β-C-H Functionalization of Amine Triggered by Trifluoromethylation of Alkene: One-Pot Synthesis of Bistrifluoromethylated Enamides and Oxazoles. Angew. Chem. Int. Ed. 2015, 54, 4041.

40. Jian Zhang, Shao-Xia Lin, Dao-Juan Cheng, Xin-Yuan Liu*, and Bin Tan*. Phosphoric Acid-Catalyzed Asymmetric Classic Passerini Reaction. J. Am. Chem. Soc.2015137, 14039.

39. Can-Liang Ma, Xiao-Long Yu, Xiao-Long Zhu, Yong-Zhou Hu, Xiao-Wu Dong, Bin Tan,* and Xin-Yuan Liu,* Platinum-Catalyzed Tandem Cyclization Reaction to Multiply Substituted Indolines under Microwave-Assisted Conditions. Adv. Synth. Catal. 2015357, 569.

38. Lin Huang, Sheng-Cai Zheng, Bin Tan,* Xin-Yuan Liu,* Trifluoromethylation-Initiated Remote Cross-Coupling of Carbonyl Compounds to Form Carbon–Heteroatom/Carbon Bonds. Chem. Eur. J. 201521, 6718. 

37. Lei Li, Jing-Yao Guo, Xing-Guo Liu, Su Chen, Yong Wang, Bin Tan,* and Xin-Yuan Liu,* Amide Groups Switch Selectivity: C–H Trifluoromethylation of α,β-Unsaturated Amides and Subsequent Asymmetric Transformation. Org. Lett. 201416, 6032.

36. Jin-Shun Lin, Xiang-Geng Liu, Xiao-Long Zhu, Bin Tan,* and Xin-Yuan Liu,* Copper-Catalyzed Aminotrifluoromethylation of Unactivated Alkenes with TMSCF3: Construction of Trifluoromethylated Azaheterocycles. J. Org. Chem. 201479, 7084.

35. Ya-Ping Xiong, Ming-Yue Wu, Xiang-Yu Zhang, Can-Liang Ma, Lin Huang, Li-Jiao Zhao, Bin Tan,* and Xin-Yuan Liu,* Direct Access to α-CF3-enones via Efficient Copper-Catalyzed Trifluoromethylation of Meyer-Schuster Rearrangement. Org. Lett. 201416, 1000.

34. Jin-Shun Lin, Ya-Ping Xiong, Can-Liang Ma, Li-Jiao Zhao, Bin Tan,* and Xin-Yuan Liu,* Efficient Copper-Catalyzed Direct Intramolecular Aminotrifluoromethylation of Unactivated Alkenes with Diverse Nitrogen-Based Nucleophiles. Chem. Eur. J. 201420, 1332.

33. Peng Yu, Jin-Shun Lin, Lei Li, Sheng-Cai Zheng, Ya-Ping Xiong, Li-Jiao Zhao, Bin Tan,* and Xin-Yuan Liu,*Enantioselective C–H Bond Functionalization Triggered by Radical Trifluoromethylation of Unactivated Alkene. Angew. Chem., Int. Ed. 201453, 11890.

32. Dao-Juan Cheng, Liang Yan, Shi-Kai Tian,* Ming-Yue Wu, Lu-Xin Wang, Zi-Li Fan, Sheng-Cai Zheng, Xin-Yuan Liu,* and Bin Tan,* Highly Enantioselective Kinetic Resolution of Axially Chiral BINAM Derivatives Catalyzed by a Brønsted Acid. Angew. Chem. Int. Ed. 201453, 3684.

31. Xing-Li Zhu, Jin-Hui Xu, Dao-Juan Cheng, Li-Jiao Zhao, Xin-Yuan Liu,* and Bin Tan,* In Situ Generation of Electrophilic Trifluoromethylthio Reagents for Enantioselective Trifluoromethylthiolation of Oxindoles. Org. Lett. 201416, 2192. 

30. Lei Li, Min Deng, Sheng-Cai Zheng, Ya-Ping Xiong, Bin Tan,* and Xin-Yuan Liu,* Metal-Free Direct Intramolecular Carbotrifluoromethylation of Alkenes to Functionalized Trifluoromethyl Azaheterocycles. Org. Lett201416, 504. 

29. Daojuan Cheng, Yoshihiro Ishihara, Bin Tan*, and Carlos F. BarbasIII*. Organocatalytic Asymmetric Assembly Reactions: Synthesis of Spirooxindoles via Organocascade Strategies. ACS Catal. 20144, 743.

28. Bin Tan, Xuan, Zhang, and Zhong, Guofu. Protecting-group directed stereospecific organocatalytic [3+2] cycloadditions: a facile access to chiral spirocyclic oxindoles. Source: Arkivoc Pages: 124-142 Published: 2014.  

27. Klaus Albertshofer, Bin Tan, and Carlos F. BarbasIII*. Asymmetric Construction of Spirocyclopentenebenzofuranone Core Structures via Highly Selective Phosphine-Catalyzed [3+2] Cycloaddition Reactions. Org. Lett. 201315, 2958.

26. Xianxing Jiang, Bin Tan, and Carlos F. Barbas III. Core-Structure-Motivated Design of Iminium-Enolate Organocascade Reactions: Enantioselective Syntheses of 5,6-Dihydroindolizines. Angew. Chem. Int. Ed. 201352, 9261.

25. Klaus Albertshofer, Bin Tan, and Carlos F. BarbasIII*. Assembly of Spirooxindole Derivatives Containing Four Consecutive Stereocenters via Organocatalytic Michael-Henry Cascade Reactions. Org. Lett. 201214, 1834.

24. Bin Tan, Xiaofei Zeng, Wendy Wen Yi Leong, Zugui Shi, Carlos F. Barbas, III,* and Guofu Zhong*. Core Structure-Based Design of Organocatalytic [3+2]-Cycloaddition Reactions: Highly Efficient and Stereocontrolled Syntheses of 3,3'-Pyrrolidonyl Spirooxindoles. Chem. Eur. J. 201218, 63.

23. Gloria Hernández-Torres, Bin Tan, and Carlos F. BarbasIII*. Organocatalysis as a Safe Practical Method for the Stereospecific Dibromination of Unsaturated Compounds. Org. Lett. 201214, 1858.

22. Bin Tan, Narihiro Toda, and Carlos F. Barbas III*. Organocatalytic Amidation and Esterification of Aldehydes with Activating Reagents by a Cross-Coupling Strategy. Angew. Chem. Int. Ed. 201251, 12538.

21. Bin Tan, Gloria Hernández-Torres,  Carlos F. Barbas III* Rationally Designed Amide Donors for Organocatalytic Asymmetric Michael Reactions. Angew. Chem. Int. Ed. 201251, 5381.

20. Bin Tan, Nuno R. Candeias, Carlos F. Barbas III. Construction of bispirooxindoles containing three quaternary stereocentres in a cascade using a single multifunctional organocatalyst. Nature Chem. 20113, 473. 

19. Bin Tan, Nuno R. Candeias, and Carlos F. BarbasIII*. Core-Structure-Motivated Design of a Phosphine-Catalyzed [3+2] Cycloaddition Reaction: Enantioselective Syntheses of Spirocyclopenteneoxindoles. J. Am. Chem. Soc. 2011133, 4672.

18. Bin Tan, Gloria Hernández-Torres, and Carlos F. BarbasIII*. Highly Efficient Hydrogen-Bonding Catalysis of the Diels-Alder Reaction of 3-Vinylindoles and Methyleneindolinones Provides Carbazolespirooxindole Skeletons. J. Am. Chem. Soc. 2011133, 12354.

17. Zugui Shi, Bin Tan, Wendy Wen Yi Leong, Xiaofei Zeng, Min Lu, and Guofu Zhong*. Catalytic Asymmetric Formal [4+1] Annulation Leading to Optically Active cis-Isoxazoline N-Oxides. Org. Lett. 201012, 5402.

16. Xiaofei Zeng, Kehan Ye, Min Lu, Pei Juan Chua, Bin Tan and Guofu Zhong*. Chiral Bronsted Acid Catalyzed Enantioselective Addition of alpha-Isocyanoacetamides to Aldehydes. Org. Lett. 201012, 2414.

15. Zhen-Jiang Xu, Di Zhu, Xiaofei Zeng, Fei Wang, Bin Tan, Yuxuan Hou, Yunbo Lva and Guofu Zhong*. Diastereoselective HOTf-catalyzed three-component one-pot 1,3-dipolar cycloaddition of alpha-diazo ester, nitrosobenzene and electron-deficient alkene. Chem. Commun. 201046, 2504.

14. Bin Tan, Yunpeng Lu, Xiaofei Zeng, Pei Juan Chua and Guofu Zhong*. Facile Domino Access to Chiral Bicyclo[3.2.1]octanes and Discovery of a New Catalytic Activation Mode. Org. Lett. 201012, 2682.

13. Pei Juan Chua, Bin Tan, Limin Yang, Xiaofei Zeng, Di Zhua and Guofu Zhong*. Highly stereoselective synthesis of indanes with four stereogenic centers via sequential Michael reaction and [3+2] cycloaddition. Chem. Commun. 201046, 7611.

12. Bin Tan, Di Zhu, Lihong Zhang, Pei Juan Chua, Xiaofei Zeng, and Guofu Zhong*. Water-More Than Just a Green Solvent: A Stereoselective One-Pot Access to All-Chiral Tetrahydronaphthalenes in Aqueous Media.45a. Bin Tan, Yunpeng Lu, Xiaofei Zeng, Pei Juan Chua and Guofu Zhong*. Chem. Eur. J. 201016, 3842.

11. Limin Yang, Bin Tan, Fei Wang and Guofu Zhong*. An Unexpected N-Heterocyclic Carbene-Catalyzed Annulation of Enals and Nitroso Compounds. Org. Chem. 200974, 1744.

10. Min Lu, Di Zhu, Yunpeng Lu, Xiaofei Zeng, Bin Tan, Zhenjiang Xu and Guofu Zhong*. Chiral Bronsted Acid-Catalyzed Enantioselective alpha-Hydroxylation of beta-Dicarbonyl Compounds. J. Am. Chem. Soc. 2009131, 4562.

9. Pei Juan Chua, Bin Tan, Xiaofei Zeng, Guofu Zhong *. L-Prolinol as a highly enantioselective catalyst for Michael addition of cyclohexanone to nitroolefins. Bioorg. Med. Chem. Lett. 200919, 3915.

8. Bin Tan, Xiaofei Zeng, Yunpeng Lu, Pei Juan Chua and Guofu Zhong*. Rational Design of Organocatalyst: Highly Stereoselective Michael Addition of Cyclic Ketones to Nitroolefins. Org. Lett. 200911, 1927.

7. Bin Tan,a Xuan Zhang,a Pei Juan Chuaa and Guofu Zhong*. Recyclable organocatalysis: highly enantioselective Michael addition of 1,3-diaryl-1,3-propanedione to nitroolefins. Chem. Commun. 200912, 779.

6. Bin Tan, Zugui Shi, Pei Juan Chua, Yongxin Li, and Guofu Zhong*.Unusual Domino Michael/Aldol Condensation Reactions Employing Oximes as N-Selective Nucleophiles Synthesis of N-Hydroxypyrroles. Angew. Chem. Int. Ed. 200948, 758.

5. Bin Tan, Pei Juan Chua, Xiaofei Zeng, Min Lu and Guofu Zhong. A highly diastereo- and enantioselective synthesis of multisubstituted cyclopentanes with four chiral carbons by the organocatalytic domino Michael-Henry reaction. Org. Lett. 200810, 3489.

4. Di Zhu, Min Lu, Pei Juan Chua, Bin Tan, Fei Wang, Xinhao Yang† and Guofu Zhong*. A Highly Stereoselective Organocatalytic Tandem Aminoxylation/Aza-Michael Reaction for the Synthesis of Tetrahydro-1,2-Oxazines. Org. Lett. 200810, 4585.

3. Bin Tan, Zugui Shi, Pei Juan Chua and Guofu Zhong. Control of four stereocenters in an organocatalytic domino double Michael reaction: Efficient synthesis of multisubstituted cyclopentanes. Org. Lett. 200810, 3425.

2. Min Lu, Di Zhu, Yunpeng Lu, Yuxuan Hou, Bin Tan, and Guofu Zhong*. Organocatalytic Asymmetric alpha-Aminoxylation/Aza-Michael Reactions for the Synthesis of Functionalized Tetrahydro-1,2-oxazines. Angew. Chem. Int. Ed. 200847, 10187.

1. Bin Tan, Pei Juan Chua, Yongxin Li and Guofu Zhong. Organocatalytic asymmetric tandem Michael-Henry reactions: A highly stereoselective synthesis of multifunctionalized cyclohexanes with two quaternary stereocenters. Org. Lett. 200810, 2437.

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